Upper Respiratory System Drugs

Upper Respiratory Disorders:
 Involves nasopharynx, pharynx, larynx, sinuses: Colds, rhinitis, sinusitis, pharyngitis
  • ANTIHISTAMINES
    • Block H1 and/or H2 receptors 
    • Side effects: Decreased SLUDGE (anticholinergic), drowsiness
    • Prototype drug: Diphenhydramine (Benadryl)—1st generation—PO, injectable (can be used for emergencies)
    • 2nd generation antihistamines: Cetirizine (Zyrtec), fexofenadine (Allegra), loratidine (Claritin)—available only by PO
  • DECONGESTANTS
    • Alpha adrenergic effects
    • Administered by nasal spray, PO
    • Drugs: Ephedrine, pseudoephedrine (Sudaphed), phenylephrine (Neo-Synephrine), oxymetazoline (Afrin)—spray
    • Side effects: Rebound congestion with overuse of spray; systemic: elevated BP, elevated blood glucose; dysrhythmias; avoid stimulants
  • INTRANASAL GLUCOCORTICOIDS
    • Systemic side effects rare; may cause nasal dryness
    • Drugs: Fluticasone (Flonase), Triamcinolone (Nasacort)
  • ANTITUSSIVES
    • Suppress cough reflex
    • Prototype drug: Dextromethorphan (Robitussin, Delsym)
        • Available OTC
        • Intoxication at high doses
  • EXPECTORANTS
    • Liquify sputum for easier production with coughing
    • Need to increase PO fluid itake
    • Drug: Guaifenesin (Robitussin, Mucinex)

No comments